Compile Data Set for Download or QSAR
maximum 50k data
Found 15 of ki for NEURONAL ACETYLCHOLINE RECEPTOR SUBUNIT ALPHA-5
having polymerids = 49000414 and
complexids = 50000439,50015332,50000420
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  0.0960nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50079456(2-Pyridin-3-yl-1-aza-bicyclo[2.2.2]octane | CHEMBL...)
Affinity DataKi:  1.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50047021(2-(6-(2-hydroxy-2-phenylethyl)-1-methylpiperidin-2...)
Affinity DataKi:  6.39nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171347(3-(Azetidin-2-ylmethoxy)-pyridine | A-85380 | CHEM...)
Affinity DataKi:  8.71nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
Affinity DataKi:  156nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86309(CAS_21019-30-7 | Methyllycaconitine | NSC_5311278)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50171341(3-Methyl-5-(1-methyl-pyrrolidin-2-yl)-isoxazole | ...)
Affinity DataKi:  803nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246823(CHEMBL4071277)
Affinity DataKi:  957nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4alpha5 nAChR expressed in HEK cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82546(CAS_14721-69-8 | MCC | N-methylcarbamylcholine | N...)
Affinity DataKi:  969nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86544(CAS_192231-16-6 | CHEMBL111580 | NSC_6442277 | SIB...)
Affinity DataKi:  991nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86543(CAS_156223-05-1 | GTS-21 | NSC_122225)
Affinity DataKi:  1.29E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Rattus norvegicus (Rat))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50246826(CHEMBL4084577)
Affinity DataKi:  1.62E+3nMAssay Description:Displacement of [3H]epibatidine from rat alpha3beta4alpha5 nAChR expressed in HEK cells after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataKi:  3.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/alpha-5/beta-4(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50446500(CHEMBL3110043)
Affinity DataKi:  9.06E+3nMAssay Description:Binding affinity to alpha3beta4alpha5 nAChR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM86241(CAS_23255-54-1 | Dihydro-Beta-erythroidine | NSC_3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed